Публикации Лаборатории Химической Трансформации Антибиотиков
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A.S. Tikhomirov, D.V. Andreeva, A.E. Shchekotikhin. Reductive elimination of alkoxy group in anthraquinone derivatives, Tetrahedron 2022, 122, 132957, https://doi.org/10.1016/j.tet.2022.132957.
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Krymov S. K., Scherbakov A.M., Dezhenkova L.G., Salnikova D.I., Solov’eva S.E., Sorokin D.V., Vullo D., De Luca V., Capasso C., Supuran C.T., Shchekotikhin A.E. Indoline-5-Sulfonamides: A Role of the Core in Inhibition of Cancer-Related Carbonic Anhydrases, Antiproliferative Activity and Circumventing of Multidrug Resistance. Pharmaceuticals, 2022, 15, 1453. https://doi.org/10.3390/ph15121453
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J.S. Chang, C.-Y. Chen, A.S. Tikhomirov, A. Islam,R.-H. Liang, C.-W. Weng, W.-H. Wu, A.E. Shchekotikhin, P.J. Chueh. Bis(chloroacetamidino)-Derived Heteroarene-Fused Anthraquinones Bind to and Cause Proteasomal Degradation of tNOX, Leading to c-Flip Downregulation and Apoptosis in Oral Cancer Cells. Cancers 2022, 14(19), 4719; https://doi.org/10.3390/cancers14194719
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Dezhenkova L.G.; Druzina A.A.; Volodina Y.L.; Dudarova N.V.; Nekrasova N.A.; Zhidkova O.B.; Grin M.A.; Bregadze V.I. Synthesis of Cobalt Bis(Dicarbollide)-Curcumin Conjugates for Potential Use in Boron Neutron Capture Therapy. Molecules 2022, 27, 4658. DOI:10.3390/molecules27144658
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Sachkova, A.A.; Andreeva, D.V.; Tikhomirov, A.S.; Scherbakov, A.M.; Salnikova, D.I.; Sorokin, D.V.; Bogdanov, F.B.; Rysina, Y.D.; Shchekotikhin, A.E.; Shchegravina, E.S.;. Fedorov A. Yu Design, Synthesis and In Vitro Investigation of Cabozantinib-Based PROTACs to Target c-Met Kinase. Pharmaceutics 2022, 14, 2829. https://doi.org/10.3390/pharmaceutics14122829
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Isagulieva, A.K.; Kaluzhny, D.N.; Beniaminov, A.D.; Soshnikova, N.V.; Shtil, A.A. Differential Impact of Random GC Tetrad Binding and Chromatin Events on Transcriptional Inhibition by Olivomycin A. International Journal of Molecular Sciences 2022, 23, 8871. https://doi.org/10.3390/ijms23168871
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M. Singh, Md.A. Haque, A.S. Tikhomirov, A.E. Shchekotikhin, U. Das, P. Kaur, Computational and Biophysical Characterization of Heterocyclic Derivatives of Anthraquinone against Human Aurora Kinase A. ACS Omega, 2022, 7, 44, 39603-39618, https://doi.org/10.1021/acsomega.2c00740
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Исагулиева А.К., Тевяшова А.Н., Штиль А.А. Антибиотики группы ауреоловой кислоты: перспективы биологически активного класса соединений. Биоорганическая химия., 2022, 48(3), 1-13. doi:10.31857/S0132342322020129
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N. Savin, A. Erofeev, V. Kolmogorov, S. Salikhov, Y. Efremov, P. Timashev, N. Grammatikova, I. Levshin, C. Edwards, Y. Korchev, P. Gorelkin. Scanning ion-conductance microscopy technique for studying the topography and mechanical properties of Candida parapsilosis yeast microorganisms; Biomaterials Science 2022. DOI:10.1039/d2bm00964a
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Олсуфьева Е.Н., Янковская В.С., Дунченко Н.И. Обзор рисков контаминации антибиотиками молочной продукции. Антибиотики и химиотерапия 2022, 67 (7–8):82-96. https://doi.org/10.37489/0235-2990-2022-67-7-8-82-96
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Щекотихин А. Е., Олсуфьева Е. Н., Янковская В. С. Антибиотики и родственные вещества. М.: Лаборатория знаний. 2022., 511 с. ISBN 978-5-93208-247-8.
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A. Shchekotikhin, V.F Traven, N.A. Pozharskaya. History and Scientific Achievements of the Department of Organic Chemistry of the Mendeleev University of Chemical Technology of Russia // in History of Organic Chemistry at Russian Universities. Eds. E. Beloglazkina, I. Beletskaya, D. Lewis, V. Nenaydenko. М.: NGB Publishing House. 2022, Р. 272-299.
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A.S. Tikhomirov, V.B. Tsvetkov, Y.L. Volodina, V.A. Litvinova, D.V. Andreeva, L.G. Dezhenkova, D.N. Kaluzhny, I.D. Treshalin, A.A. Shtil, A.E. Shchekotikhin. Heterocyclic ring expansion yields anthraquinone derivatives potent against multidrug resistant tumor cells, Bioorganic Chemistry, 2022, 127, 105925, https://doi.org/10.1016/j.bioorg.2022.105925
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E. Di Giorgio, A. Ferino, H. Choudhary, P. M.G. Löffler, F. D'Este, V. Rapozzi, A. Tikhomirov, A. Shchekotikhin, S. Vogel, L.E. Xodo. Photosensitization of pancreatic cancer cells by cationic alkyl-porphyrins in free form or engrafted into POPC liposomes: The relationship between delivery mode and mechanism of cell death, Journal of Photochemistry and Photobiology B: Biology, 2022, 231, 112449, https://doi.org/10.1016/j.jphotobiol.2022.112449
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Levshin I.B., Simonov A.Y., Lavrenov S.N., Panov A.A., Grammatikova N.E., Alexandrov A.I., Ghazy E.S.M.O., Savin N.A., Gorelkin P.V., Erofeev A.S., Polshakov V.I. Antifungal Thiazolidines: Synthesis and Biological Evaluation of Mycosidine Congeners. Pharmaceuticals, 2022, 15, 5, 563-586. DOI: 10.3390/ph15050563
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Treshchalin M.I., Polozkova V.A., Moiseenko E.I., Treshalina H.M., Shchekotikhin A.E., Pereverzeva E.R. Evaluation of Toxic Properties of New Glycopeptide Flavancin on Rats. Pharmaceuticals, 2022, 15, 661. DOI: 10.3390/ph15060661
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Buravchenko G.I. Maslov D.A., Alam M.S., Grammatikova N.E., Frolova S.G., Vatlin A.A., Tia, X., Ivanov I.V., Bekker O.B., Kryakvin M.A., Dontsova O.A., Danilenko V.N., Zhang T., Shchekotikhin A.E. Synthesis and Characterization of Novel 2-Acyl-3-trifluoromethylquinoxaline 1,4-Dioxides as Potential Antimicrobial Agents. Pharmaceuticals 2022, 15(2), 155, https://doi.org/10.3390/ph15020155
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M.H. Lin, A. Islam, Y.-H. Liu, C.-W. Weng, J.-H. Zhan, R.-H. Liang, A.S. Tikhomirov, A.E. Shchekotikhin, P.J. Chueh, Antibiotic heliomycin and its water-soluble 4-aminomethylated derivative provoke cell death in T24 bladder cancer cells by targeting sirtuin 1 (SIRT1). American Journal of Cancer Research 2022, 12(3), 1042-1055, www.ajcr.us /ISSN:2156-6976/ajcr0140356
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Perera W.H., Scherbakov A.M., Buravchenko G.I., Mikhaevich E.I., Guimar S., Cos P., Shchekotikhin A.E., Monzote L., Setzer W.N. In Vitro Pharmacological Screening of Essential Oils from Baccharis parvidentata and Lippia origanoides Growing. Molecules, 2022, 27, 1926, https://doi.org/10.3390/molecules27061926