Публикации Лаборатории Химической Трансформации Антибиотиков

 

  1. A.S. Tikhomirov, D.V. Andreeva, A.E. Shchekotikhin. Reductive elimination of alkoxy group in anthraquinone derivatives, Tetrahedron 2022, 122, 132957, https://doi.org/10.1016/j.tet.2022.132957. 

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  2. Krymov S. K., Scherbakov A.M., Dezhenkova L.G., Salnikova D.I., Solov’eva S.E., Sorokin D.V., Vullo D., De Luca V., Capasso C., Supuran C.T., Shchekotikhin A.E. Indoline-5-Sulfonamides: A Role of the Core in Inhibition of Cancer-Related Carbonic Anhydrases, Antiproliferative Activity and Circumventing of Multidrug Resistance. Pharmaceuticals, 2022, 15, 1453. https://doi.org/10.3390/ph15121453

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  3. J.S. Chang, C.-Y. Chen, A.S. Tikhomirov, A. Islam,R.-H. Liang, C.-W. Weng, W.-H. Wu, A.E. Shchekotikhin, P.J. Chueh. Bis(chloroacetamidino)-Derived Heteroarene-Fused Anthraquinones Bind to and Cause Proteasomal Degradation of tNOX, Leading to c-Flip Downregulation and Apoptosis in Oral Cancer Cells. Cancers 2022, 14(19), 4719; https://doi.org/10.3390/cancers14194719

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  4. Dezhenkova L.G.; Druzina A.A.; Volodina Y.L.; Dudarova N.V.; Nekrasova N.A.; Zhidkova O.B.; Grin M.A.; Bregadze V.I. Synthesis of Cobalt Bis(Dicarbollide)-Curcumin Conjugates for Potential Use in Boron Neutron Capture Therapy. Molecules 2022, 27, 4658. DOI:10.3390/molecules27144658

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  5. Sachkova, A.A.; Andreeva, D.V.; Tikhomirov, A.S.; Scherbakov, A.M.; Salnikova, D.I.; Sorokin, D.V.; Bogdanov, F.B.; Rysina, Y.D.; Shchekotikhin, A.E.; Shchegravina, E.S.;. Fedorov A. Yu Design, Synthesis and In Vitro Investigation of Cabozantinib-Based PROTACs to Target c-Met Kinase. Pharmaceutics 2022, 14, 2829. https://doi.org/10.3390/pharmaceutics14122829

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  6. Isagulieva, A.K.; Kaluzhny, D.N.; Beniaminov, A.D.; Soshnikova, N.V.; Shtil, A.A. Differential Impact of Random GC Tetrad Binding and Chromatin Events on Transcriptional Inhibition by Olivomycin A. International Journal of Molecular Sciences 2022, 23, 8871. https://doi.org/10.3390/ijms23168871

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  7. M. Singh, Md.A. Haque, A.S. Tikhomirov, A.E. Shchekotikhin, U. Das, P. Kaur, Computational and Biophysical Characterization of Heterocyclic Derivatives of Anthraquinone against Human Aurora Kinase A. ACS Omega, 2022, 7, 44, 39603-39618, https://doi.org/10.1021/acsomega.2c00740

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  8. Исагулиева А.К., Тевяшова А.Н., Штиль А.А. Антибиотики группы ауреоловой кислоты: перспективы биологически активного класса соединений. Биоорганическая химия., 2022, 48(3), 1-13. doi:10.31857/S0132342322020129

  9. N. Savin, A. Erofeev, V. Kolmogorov, S. Salikhov, Y. Efremov, P. Timashev, N. Grammatikova, I. Levshin, C. Edwards, Y. Korchev, P. Gorelkin. Scanning ion-conductance microscopy technique for studying the topography and mechanical properties of Candida parapsilosis yeast microorganisms; Biomaterials Science 2022. DOI:10.1039/d2bm00964a

  10. Олсуфьева Е.Н., Янковская В.С., Дунченко Н.И. Обзор рисков контаминации антибиотиками молочной продукции. Антибиотики и химиотерапия 2022, 67 (7–8):82-96. https://doi.org/10.37489/0235-2990-2022-67-7-8-82-96

  11. Щекотихин А. Е., Олсуфьева Е. Н., Янковская В. С. Антибиотики и родственные вещества. М.: Лаборатория знаний. 2022., 511 с. ISBN 978-5-93208-247-8.

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  12. A. Shchekotikhin, V.F Traven, N.A. Pozharskaya. History and Scientific Achievements of the Department of Organic Chemistry of the Mendeleev University of Chemical Technology of Russia // in History of Organic Chemistry at Russian Universities. Eds. E. Beloglazkina, I. Beletskaya, D. Lewis, V. Nenaydenko. М.: NGB Publishing House. 2022, Р. 272-299.

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  13. A.S. Tikhomirov, V.B. Tsvetkov, Y.L. Volodina, V.A. Litvinova, D.V. Andreeva, L.G. Dezhenkova, D.N. Kaluzhny, I.D. Treshalin, A.A. Shtil, A.E. Shchekotikhin. Heterocyclic ring expansion yields anthraquinone derivatives potent against multidrug resistant tumor cells, Bioorganic Chemistry, 2022, 127, 105925, https://doi.org/10.1016/j.bioorg.2022.105925

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  14. E. Di Giorgio, A. Ferino, H. Choudhary, P. M.G. Löffler, F. D'Este, V. Rapozzi, A. Tikhomirov, A. Shchekotikhin, S. Vogel, L.E. Xodo. Photosensitization of pancreatic cancer cells by cationic alkyl-porphyrins in free form or engrafted into POPC liposomes: The relationship between delivery mode and mechanism of cell death, Journal of Photochemistry and Photobiology B: Biology, 2022, 231, 112449, https://doi.org/10.1016/j.jphotobiol.2022.112449

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  15. Levshin I.B., Simonov A.Y., Lavrenov S.N.,  Panov A.A., Grammatikova N.E., Alexandrov A.I., Ghazy E.S.M.O., Savin N.A., Gorelkin P.V., Erofeev A.S., Polshakov V.I. Antifungal Thiazolidines: Synthesis and Biological Evaluation of Mycosidine Congeners. Pharmaceuticals, 2022, 15, 5, 563-586. DOI: 10.3390/ph15050563

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  16. Treshchalin M.I., Polozkova V.A., Moiseenko E.I., Treshalina H.M., Shchekotikhin A.E., Pereverzeva E.R. Evaluation of Toxic Properties of New Glycopeptide Flavancin on Rats. Pharmaceuticals, 2022, 15, 661. DOI: 10.3390/ph15060661

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  17. Buravchenko G.I. Maslov D.A., Alam M.S., Grammatikova N.E., Frolova S.G., Vatlin A.A., Tia, X., Ivanov I.V., Bekker O.B., Kryakvin M.A., Dontsova O.A., Danilenko V.N., Zhang T., Shchekotikhin A.E. Synthesis and Characterization of Novel 2-Acyl-3-trifluoromethylquinoxaline 1,4-Dioxides as Potential Antimicrobial Agents. Pharmaceuticals 2022, 15(2), 155, https://doi.org/10.3390/ph15020155

  18. M.H. Lin, A. Islam, Y.-H. Liu, C.-W. Weng, J.-H. Zhan, R.-H. Liang, A.S. Tikhomirov, A.E. Shchekotikhin, P.J. Chueh, Antibiotic heliomycin and its water-soluble 4-aminomethylated derivative provoke cell death in T24 bladder cancer cells by targeting sirtuin 1 (SIRT1). American Journal of Cancer Research 2022, 12(3), 1042-1055, www.ajcr.us /ISSN:2156-6976/ajcr0140356

  19. Perera W.H., Scherbakov A.M., Buravchenko G.I., Mikhaevich E.I., Guimar S., Cos P., Shchekotikhin A.E., Monzote L., Setzer W.N. In Vitro Pharmacological Screening of Essential Oils from Baccharis parvidentata and Lippia origanoides Growing. Molecules, 2022, 27, 1926, https://doi.org/10.3390/molecules27061926

  20. Buravchenko G.I., Scherbakov A.M., Dezhenkova L.G., Fidalgo L., Shchekotikhin, A.E. Synthesis of 7-Amino-6-Halogeno-3-Phenylquinoxaline-2-Carbonitrile 1,4-Dioxides: A Way Forward for Targeting Hypoxia and Drug Resistance of Cancer Cells, RSC Advances, 2021, 11, 38782, doi:10.1039/d1ra07978f.

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  21. Krymov S.K., Scherbakov A.M., Salnikova D.I., Sorokin D.V., Dezhenkova L.G., Ivanov I.V., Vullo D., De Luca V., Capasso C., Supuran C.T., Shchekotikhin A.E., Synthesis, biological evaluation, and in silico studies of potential activators of apoptosis and carbonic anhydrase inhibitors on isatin-5-sulfonamide scaffold. European Journal of Medicinal Chemistry, 2021, 228, 113997, https://doi.org/10.1016/j.ejmech.2021.113997

  22. Тевяшова А.Н., Шаповалова К.С. Потенциал разработки аминогликозидных антибиотиков нового поколения. Химико-фармацевтический журнал 2021, 55, 7–23 https://doi.org/10.30906/0023-1134-2021-55-9-7-23 

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  23. Omelchuk O.A., Malyshev V.I., Medvedev M.G., Lysenkova L.N., Belov N.M., Dezhenkova L.G., Grammatikova N.E., Scherbakov A.M., Shchekotikhin A.E. Stereochemistries and Biological Properties of Oligomycin A Diels–Alder Adducts. Journal of Organic Chemistry 2021, 86, 12, 7975–7986. DOI: 10.1021/acs.joc.1c00296.

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  24. Scherbakov A.M., Sorokin D.V., Omelchuk O.A., Shchekotikhin A.E., Krasil'nikov M.A. Glucose starvation greatly enhances antiproliferative and antiestrogenic potency of oligomycin A in MCF-7 breast cancer cells. Biochimie 2021, 186, 51–58. DOI: 10.1016/j.biochi.2021.04.003.

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  25. Volodina Y.L., Tikhomirov A.S., Dezhenkova L.G., Ramonova A.A., Kononova A. V., Andreeva D. V., Kaluzhny D.N., Schols D., Moisenovich M.M., Shchekotikhin A.E., Shtil A.A. Thiophene-2-carboxamide derivatives of anthraquinone: A new potent antitumor chemotype. European Journal of Medicinal Chemistry 2021, № 221, 113521. DOI: 10.1016/j.ejmech.2021.113521.

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  26. Tikhomirov A.S., Abdelhamid M.A.S., Nadysev G.Y., Zatonsky G.V., Bykov E.E., Chueh P.J., Waller Z.A.E., Shchekotikhin A.E. Water-Soluble Heliomycin Derivatives to Target i-Motif DNA. Journal of Natural Products 2021, 84(5), 1617-1625. doi:10.1021/acs.jnatprod.1c00162.

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  27. Moiseenko E.I., Erdei R., Grammatikova N.E., Mirchink E.P., Isakova E.B., Pereverzeva E.R., Batta G., Shchekotikhin A.E. Aminoalkylamides of Eremomycin Exhibit an Improved Antibacterial Activity. Pharmaceuticals 2021, 14(4), 379. doi:10.3390/ph14040379.

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  28. Blokhina S.V., Ol'khovich M. V., Sharapova A. V., Levshin I. B., Perlovich G. L. Study of dissolution and transfer processes of new bioactive thiazolo[4,5-d]pyrimidine derivatives in modeling biological systems. Journal of Molecular Liquids 2021, 337, 116395. doi:10.1016/j.molliq.2021.116395

  29. Volkova T. V., Simonova O. R., Levshin I. B., Perlovich G.L. Physicochemical profile of new antifungal compound: pH-dependent solubility, distribution, permeability and ionization assay. Journal of Molecular Liquids 2021, 116535 doi.org/10.1016/j.molliq.2021.116535.

  30. Blokhina S. V., Sharapova A. V., Ol'khovich M. V., Doroshenko I. A., Levshin I. B., Perlovich G. L. (). Synthesis and antifungal activity of new hybrids thiazolo[4,5-d]pyrimidines with (1H-1,2,4)triazole. Bioorganic and Medicinal Chemistry Letters 2021, 40, 127944. doi.org/10.1016/j.bmcl.2021.127944

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  31. Izsépi L., Erdei R., Tevyashova A.N., Grammatikova N.E., Shchekotikhin A.E., Herczegh P., Batta G. Bacterial cell wall analogue peptides control the oligomeric states and activity of the glycopeptide antibiotic Eremomycin: solution NMR and antimicrobial studies. Pharmaceuticals 2021, 14(2), 83; https://doi.org/10.3390/ph14020083

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  32. Тевяшова А.Н., Чудинов М.В. Прогресс в медицинской химии органических соединений бора. Успехи химии 2021, 90(4), 451–487; https://doi.org/10.1070/RCR4977

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  33. Tevyashova A.N. Recent trends in synthesis of chloramphenicol new derivatives. Antibiotics 2021, 10, 370 https://doi.org/10.3390/antibiotics10040370

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  34. Litvinova V.А., Tikhomirov A.S. New methods for synthesis of 1-benzothiophene-3-carboxylic acid derivatives (microreview). Chemistry of Heterocycic Compounds 2021, 57(2), 131–133. DOI: https://doi.org/10.1007/s10593-021-02882-x.

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  35. Singh M., Malhotra L., Haque M.A., Kumar M., Tikhomirov A.S, Litvinova V. A, Korolev A.M., Ethayathulla A.S., Das U., Shchekotikhin A.E., Kaur P. Heteroarene-fused anthraquinone derivatives as potential modulators for human aurora kinase B. Biochimie 2021, 182, 152-165. DOI: https://doi.org/10.1016/j.biochi.2020.12.024

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  36. Buravchenko G.I., Scherbakov A.M., Dezhenkova L.G., Bykov E.E., Solovieva S.E., Korlukov A.A., Sorokin D.V., Monzote Fidalgo L, Shchekotikhin A.E. Discovery of derivatives of 6(7)-amino-3-phenylquinoxaline-2-carbonitrile 1,4-dioxides: novel, hypoxia-selective HIF-1α inhibitors with strong antiestrogenic potency. Bioorganic Chemistry 2020, 104, 104324, doi: 10.1016/j.bioorg.2020.104324.p1

     

  37. Monzote L., Scherbakov A.M., Scull R., Satyal P., Cos P., Shchekotikhin A.E., Gille L., Setzer W.N. Essential Oil from Melaleuca leucadendra: Antimicrobial, Antikinetoplastid, Antiproliferative and Cytotoxic Assessment. Molecules 2020, 25, 5514, doi: 10.3390/molecules25235514.p2

     

  38. Monzote L., Scherbakov A. M., Scull R., Gutierrez Y. I., Satyal P., Cos P., Shchekotikhin A. E., Gille L., Setzer W. N. Pharmacological Assessment of the Carvacrol Chemotype Essential Oil From Plectranthus amboinicus Growing in Cuba. Natural Product Communications 2020, 15, № 10, 1–12, DOI: 10. 1177/ 1934 578X 20962233.p3
  39. Моисеенко Е. И., Грамматикова Н. Э., Щекотихин А. Е. Синтез и антибактериальная активность аминоалкиламидов эремомицина. Макрогетероциклы 2020, Т. 13, № 3, 298-304, DOI: 10.6060/mhc200812s p4

     

  40. Lavrenov S.N., Isakova E.B., Panov A.A., Simonov A.Y., Tatarsky V.V., Trenin A.S. N-(Hydroxyalkyl) Derivatives of tris(1H-indol-3-yl)methylium salts as promising antibacterial agents: Synthesis and biological evaluation. Pharmaceuticals 2020, 13 (12), 469, https://doi.org/10.3390/ph13120469p5

     

  41. Bespyatykh J., Bespiatykh D., Malakhova M., Klimina K., Bespyatykh A., Varizhuk A., Tevyashova A., Nikolenko T., Pozmogova G., Ilina E., Shitikov E. Aureolic Acid Group of Agents as Potential Antituberculosis Drugs. Antibiotics 2020, 9(10), 715-730. DOI: 10.3390/antibiotics9100715p6

     

  42. D.V. Andreeva, A.S. Tikhomirov, A.E. Shchekotikhin. Ligands of G-quadruplex nucleic acids, Russian Chemical Reviews 2021, 90(1), 1-38, DOI: 10.1070/RCR4968p7

     

  43. Shchegravina E.S., Svirshchevskay E.V., Combes S., Allegro D., Barbier P., Gigant B., Varela P.F., Gavryushin A.E., Kobanova D.A., Shchekotikhin A.E., Fedorov A.Yu. Discovery of dihydrofuranoallocolchicinoids - Highly potent antimitotic agents with low acute toxicity. European Journal of Medicinal Chemistry, 2020, 207, 112724. doi: 10.1016/j.ejmech.2020.112724. 1

     

  44. Popov A., Klimovich A., Styshova O., Moskovkina T., Shchekotikhin A., Grammatikova N., Dezhenkova L., Kaluzhny D., Deriabin P., Gerasimenko A., Udovenko A., Stonik V. Design, synthesis and biomedical evaluation of mostotrin, a new water soluble tryptanthrin derivative. International Journal of Molecular Medicine, 2020, 46(4), P. 1335-1346. DOI: 10.3892/ijmm.2020.4693 2

     

  45. Litvinova V.A., Tikhomirov A.S., Ivanov I.V., Solovieva S.E., Shchekotikhin A.E. A facile access to 2-substituted naphtho[2,3-g]quinoline-3-carboxylic acid esters via intramolecular cyclization and PyBOP-promoted functionalization. Tetrahedron, 2020, 76(36), 131418. https://doi.org/10.1016/j.tet.2020.131418  3

     

  46. Andreeva D.V., Tikhomirov A.S., Dezhenkova L.G., Kaluzhny D.N., Mamaeva O.K., Solovyova S.E., Sinkevich Y.B., Shchekotikhin A.E. Heterocyclic analogs of 5,12-naphthacenequinone 16. Synthesis and properties of new DNA ligands based on 4,11-diaminoanthra[2,3-b]thiophene-5,10-dione. Chemistry of Heterocyclic Compounds, 2020, 56(6), 727–733, DOI: 10.1007/s10593-020-02723-3 

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  47. Vasin A.G., Dezhenkova L.G., Ivanov I.V., Scherbakov A.M., Shchekotikhin A.E. Synthesis and antiproliferative activity of salicylidenehydrazones based on indole-2(3)-carboxylic acids. Chemistry of Heterocyclic Compounds, 2020, 56(6), 734–740, DOI: 10.1007/s10593-020-02724-2  5

     

  48. Lavrenov S.N., Bychkova O.P., Dezhenkova L.G., Mkrtchyan A.S., Tatarskiy V.V., Tsvigun E.A., Trenin A.S. Synthesis and study of cytotoxic activity of novel 3,3-bis(indol-3-yl)-1,3-dihydroindol-2-ones. Chemistry of Heterocyclic Compounds, 2020, 56(6), Р.741–746, DOI: 10.1007/s10593-020-02725-1  6
  49. Tevyashova A.N. Oxaborine derivatives: synthesis and therapeutic potential (minireview). Chemistry of Heterocyclic Compounds, 2020, 56 (6), 715–718. https://doi.org/10.1007/s10593-020-02720-6 7

     

  50. Tevyashova A.N., Bychkova E.N., Solovieva S.E., Zatonsky G.V., Grammatikova N.E., Isakova E.B., Mirchink E.P., Treshchalin I.D., Pereverzeva E.R., Bykov E.E., Efimova S.S., Ostroumova O.S., Shchekotikhin A.E. Discovery of Amphamide, a Drug Candidate for the Second Generation of Polyene Antibiotics. ACS Infectious Diseases, 2020, 6, 2029−2044 https://dx.doi.org/10.1021/acsinfecdis.0c00068  8

     

  51. Beniaminov A.D., Chashchina G.V., Livshits M.A., Kechko O.I., Mitkevich V.A., Mamaeva O.K., Tevyashova A.N., Shtil A.A., Shchyolkina A.K., Kaluzhny D.N. Discrimination between G/C Binding Sites by Olivomycin A Is Determined by Kinetics of the Drug-DNA Interaction. International Journal of Molecular Sciences, 2020, 21(15), 5299 https://doi.org/10.3390/ijms21155299 9

     

  52. Kuliabina E.V., Tevyashova A.N., Solov’eva S.E., Melkova O.N., Guskova E.A. Reference Materials of Composition of Biologically Active Substances. Measurement Techniques, 2020, 63(4), 325-331 https://doi.org/10.1007/s11018-020-01790-4. 10

     

  53. Tikhomirov A.S., Litvinova V.A., Andreeva D.V., Tsvetkov V.B., Dezhenkova L.G., Volodina Y.L., Kaluzhny D.N.,Treshalin I.D., Schols D. Ramonova A.A., Moisenovich M.M., Shtil A.A., Shchekotikhin A.E. Amides of pyrrole- and thiophene-fused anthraquinone derivatives: A role of the heterocyclic core in antitumor properties. European Journal of Medicinal Chemistry, 2020, 199, 112294. https://doi.org/10.1016/j.ejmech.2020.112294.mm1

     

  54. Sagnou M., Novikov F.N., Ivanova E.S., Alexiou P., Stroylov V.S., Titov I.Y., Tatarskiy V.V., Vagida M. S., Pelecanou M., Shtil A.A., Chilov G.G. Novel curcumin derivatives as P-glycoprotein inhibitors: Molecular modeling, synthesis and sensitization of multidrug resistant cells to doxorubicin. European Journal of Medicinal Chemistry, 2020, 198, 112331, https://doi.org/10.1016/j.ejmech.2020.112331m2
  55. Shchekotikhin A.E., Treshalina H.M., Treshchalin M.I., Pereverzeva E.R.,Isakova H.B., Tikhomirov A.S. Experimental Evaluation of Anticancer efficiency and acute toxicity of anthrafuran for oral administration, Pharmaceuticals 2020, 13(5), 81, https://doi.org/10.3390/ph13050081mm

  56. Vatlin A.A., Bekker O.B., Lysenkova L.N., Shchekotikhin A.E., Danilenko V.N. Bioinformatics Analysis of Genes of Streptomyces Xinghaiensis (Fradiae) ATCC 19609 With a Focus on Mutations Conferring Resistance to Oligomycin A and Its Derivatives. Journal of Global Antimicrobial Resistance, 2020, 22, 47-53. doi:10.1016/j.jgar.2020.01.026.

  57. Buravchenko G.I., Scherbakov А.M., Korlukov A.А., Dorovatovskii P.V., Shchekotikhin A.E. Revision of the regioselectivity of the Beirut reaction of monosubstituted benzofuroxans with benzoylacetonitrile. 6-Substituted quinoxaline-2-carbonitrile 1,4-dioxides: structural characterization and estimation of anticancer activity and hypoxia selectivity. Current Organic Chemistry, 2020, 17, 1-11, DOI: 10.2174/1570179416666191210100754g1
  58. Ferino A., Nicoletto G., D’Este F. Zorzet S., Lago S., Richter S.N., Tikhomirov A., Shchekotikhin A., Xodo L.E. Photodynamic therapy for ras-driven cancers: targeting g-quadruplex RNA structures with bifunctional alkyl-modified porphyrins. Journal of Medicinal Chemistry, 2020, 63(3), 1245-1260. https://doi.org/10.1021/acs.jmedchem.9b01577g2
  59. Olsufyeva E.N., Yankovskaya V.S., Main trends in the design of semi-synthetic antibiotics of a new generation, Russian Chemical Reviews, 2020, 89(3), 339–378. DOI: https://doi.org/10.1070/RCR4892 g3

     

  60. A.S. Tikhomirov, I.V. Ivanov, A.M. Korolev, A.E. Shchekotikhin. β-Hydroxylation of anthraquinone derivatives with benzaldehyde oxime as a source of hydroxyl group. Tetrahedron, 2019, 75, 130623. https://doi.org/10.1016/j.tet.2019.130623
     

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  61. Panov A.A., Lavrenov S.N., Simonov A.Yu., Mirchink E.P., Isakova E.., Trenin A.S. // Synthesis and antimicrobial activity of 3,4-bis(arylthio)maleimides. /J. Antibiot (Tokyo). 2019. V. 71. № 2. P. 122-124. DOI : 10.1038/s41429-018-0122-3.
     

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  62. Tevyashova A.N., Korolev A.M., Mirchink E.P., Isakova E.B., Osterman I.A. //Synthesis and evaluation of biological activity of benzoxaborole derivatives of azithromycin. / J. Antibiot (Tokyo). 2019. V. 72. № 1. Р.22-33. DOI: 10.1038/s41429-018-0107-2
     

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  63. Tevyashova A.N., Bychkova E.N., Korolev A.M., Isakova E.B., Mirchink E.P., Osterman I.A., Erdei R., Szucs. Z., Bata G. // Synthesis and evaluation of biological activity for dual-acting antibiotics on the basis of azithromycin and glycopeptides./ Bioorganic&MedicinalChemistry Letters 2019. V. 29. № 2. P. 276-280. DOI: 10.1016/j.bmcl.2018.11.038 WOS Q2
     

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  64. Sergeev A.V., Tevyashova A.N., Vorobyov A.P., Gromova, E.S. // The Effect of Antitumor Antibiotic Olivomycin A and Its New Semi-synthetic Derivative Olivamide on the Activity of Murine DNA Methyltransferase Dnmt3a./ Biochemistry (Moscow). 2019. V. 84. № 1. P. 62-70. DOI: 10.1134/S0320972519020064

  65. Bekker O.B., Vatlin A.A., Zakharevich N.V., Lysenkova L.N., Shchekotikhin A.E., Danilenko V.N.// Draft Genome Sequence of Streptomyces xinghaiensis (fradiae) OlgR, a Strain Resistant to Oligomycin A./ Microbiol Resour Announc. 2019. V. 8. № 2. № статьи: e01531-18. DOI: 10.1128/MRA.01531-18.

  66. Моисеенко Е.И., Грамматикова Н.Э., Щекотихин А. Е.// Пиколиламиды эремомицина и катионные липогликопептиды на их основе: cинтез и оценка антимикробных свойств./ Макрогетероциклы, 2019. Т. 12. №1. С. 98-106. DOI: 10.6060/mhc181216s

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  74. Evgenia N. Olsufyeva, Andrey E. Shchekotikhin, Elena N. Bychkova, Eleonora R. Pereverzeva, Ivan D. Treshalin, Elena P. Mirchink1, Elena B. Isakova, Mikhail G. Chernobrovkin, Roman S. Kozlov, Andrey V. Dekhnich, Maria N. Preobrazhenskaya Eremomycin pyrrolidide: a novel semisynthetic glycopeptide with improved chemotherapeutic properties Drug Design, Development and Therapy 2018:12 1–11Eremomycin
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  88.     A.S. Tikhomirov, V.A. Litvinova, Y.N. Luzikov, A.M. Korolev, Y.B. Sinkevich, A.E. Shchekotikhin. Heterocyclic analogs of 5,12-naphtacenequinone 14. Synthesis of naphto[2,3-f]indole-3-carboxylic acid derivatives. Chemistry of Heterocyclic Compounds. 2017. № 10, 1072-1079.Chem of heterocyclic compaunds
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  94.     Grinberg V.Y., Tsvetkov V.B., Markova A.A., Dezhenkova L.G., Burova T.V., Grinberg N.V., Dubovik A.S., Plyavnik N.V., Shtil A.A. Interactions of non-phosphorous glycerolipids with DNA: Energetics, Molecular docking and topoisomerase I attenuation. Anti-Cancer Agents in Medicinal Chemistry. 2016. V.16, Р.335-346.
  95.     Chang J., Zhou H., Preobrazhenskaya M., Tao P., Kim S.J. The сarboxyl terminus of eremomycin facilitates binding to the non D-Ala-D-Ala segment of the peptidoglycan pentapeptide stem. Biochemistry. 2016. V.55, №24, Р.3383–3391.
  96.     Принцевская С.С., Королев А.М., Исакова E.Б., Мирчинк E.П., Тевяшова А.Н. Гибридные антибиотики на основе азитромицина и гликопептидов – синтез и антибактериальная активность. Антибиотики и химиотерапия 2016. Т.61, №11-12
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  98.     M. Singh, S,J. Kim, S. Sharif, M. Preobrazhenskaya, J. Schaefer..REDOR constraints on the peptidoglycan lattice architecture of Staphylococcus aureus and its FemA mutant Biochimica et Biophysica Acta (BBA) - Biomembranes (Available online 2 June 2014) DOI:10.1016/j. bbamem.2014.05.
  99.     Printsevskaya SS, Reznikova MI, Korolev AM, Lapa GB, Olsufyeva EN, Preobrazhenskaya MN, Plattner JJ, Zhang YK Synthesis and study of antibacterial activities of antibacterial glycopeptide antibiotics conjugated with benzoxaboroles. Future Med Chem.(2013) Apr;5(6):641-52, ИФ-3,31
  100.     Лапчинская О.А.., Погожева В.В., Пономаренко В.И., Федорова Г.Б., Катруха Г.С., Преображенская М.Н. Штамм Streptomyces griseocarneus subsp. Bleomycini ВКПМ-S887 – продуцент блеомицина А2 и способ получения антибиотика блеомицина А2 Патент на изобретение № 2355758 приоритет от 27 апреля 2007 г
  101.     Sung Joon Kim, Lynette Cegelski, Maria Preobrazhenskaya, and Jacob Schaefer Structures of Staphylococcus aureus cell-wall complexes with vancomycin, eremomycin, and chloroeremomycin derivatives by 13C{19F} and 15N{19F} rotational-echo double resonance Biochemistry. 2006; 45, № 16, 5235-50
  102.     Kirk R. Maples1, Conrad Wheeler, Emily Ip, Jake Plattner, Daniel Chu Maria N. Preobrazhenskaya, Svetlana S. Printsevskaya, Svetlana E. Solovieva, Evgenia N. Olsufyeva, Henry Heine, Julie Lovchik and C. Richard Lyons A Novel Semisynthetic Derivative of Antibiotic Eremomycin Active against Drug-resistant Gram-positive Pathogens Including Bacillus anthracis J. Med.Chem. 2007, # 15, P.p.3681-3685
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  104.     Jan Balzarini,Els Keyaertsa, Leen Vijgena, Herman Egberink, Erik De Clercq, Marc Van Ransta, Svetlana S. Printsevskaya, Eugenia N. Olsufyeva, Svetlana E. Solovieva, Maria N. Preobrazhenskaya Inhibition Of Feline (Fipv) And Human (Sars) Coronavirus By Semisynthetic Derivatives Of Glycopeptide Antibiotics Antiviral Res 2006, v 72(1), 20-33
  105.     Maria N. Preobrazhenskaya and Eugenia N. Olsufyeva Polycyclic Peptide And Glycopeptide Antibiotics And Their Derivatives As Inhibitors Of Hiv Entry Antiviral Research 2006 v. 71, #2-3, pp 227-236
  106.     S. S. Printsevskaya, S. E. Solovieva, E. N. Olsufyeva, E. P. Mirchink, E. B. Isakova, E. De Clercq, J. Balzarini & M. N. Preobrazhenskaya. Structure-Activity relationships studies on a series of antiviral and antibacterial aglycon derivatives of the glycopeptide antibiotics vancomycin, eremomycin and dechloroeremomycin. J. Med. Chem. 2005. 48, 3885-3890
  107.     Svetlana S. Printsevskaya, Svetlana E. Solovieva#, Evgenia N. Olsufyeva#, Elena P. Mirchink, Elena B. Isakova#, Erik De Clercq, Jan Balzarini & Maria N. Preobrazhenskaya Structure-Activity Relationship Studies of a Series of Antiviral and Antibacterial Aglycon Derivatives of the Glycopeptide Antibiotics Vancomycin, Eremomycin, and Dechloroeremomycin J. Med. Chem.; 2005; 48(11) pp 3885 – 3890)
  108.     S.I. Maffioli, R. Ciabatti, G. Romanò, E. Marzorati, M. Preobrazhenskaya and A. Pavlov Synthesis and antibacterial activity of alkyl derivatives of the glycopeptide antibiotic A40926 and their amides Bioorganic & Medicinal Chemistry Letters Vol 15/16 pp 3801-3805
  109.     Maria N. Preobrazhenskaya, Svetlana S. Printsevskaya, Eugenia N. Olsufyeva, Svetlana Solovieva, Erik De Clercq, Jan Balzarini Derivatives of glycopeptide antibiotics with antiviral activities Drugs of the Future, 2004, 29 (Suppl. A) XVIII th Int. Symp. On MEDICINAL CHEMISTRY, p 375, 2004
  110.     Maria Preobrazhenskaya, Erik De Clercq,Jan Balzarini Glycopeptide antibiotic derivatives Patent filed on Sept. 1, 2003 with application n° PCT/BE03/00144 WO 2004/019970 A2 , August 30, 2002 Publication date 11 March 2004
  111.     Maria N.Preobrazhenskaya† and Eugenia N.Olsufyeva Patents on Glycopeptides of Vancomycin Family and Their Derivatives as Antimicrobials: January 1999 – June 2003* Expert Opinion Ther. Patents (2004) 14 (2):141-173
  112.     Irina S. Severina,Natalya V. Pyatakova,Alexander B. Postnikov,Maria N. Preobrazhenskaya,Yuri V. Khropov Antitumour antibiotic streptonigrin and its derivatives as the inhibitors of nitric oxide-dependent activation of soluble guanylate cyclase European Journal of Pharmacology 483 (2004), 127-132
  113.     M.N.Preobrazhenskaya and Eugenia N.Olsufyeva. Patents on Glycopeptides of Vancomycin Family and Their Derivatives as Antimicrobials: January 1999 - June 2003*. Expert Opinion Ther. Patents (2004) 14 (2):141-173
  114.     S. S. Printsevskaya, A.Y. Pavlov, E. N. Olsufyeva, E. P. Mirchink, and M. N. Preobrazhenskaya. The role of the glycopeptide framework in the antibacterial activity of hydrophobic derivatives of glycopeptide antibiotics. J. Med. Chem. 2003, 46, 1204-1209
  115.     J.Balzarini, Ch. Pannecouque, E. De Clercq,A.Y. Pavlov, S. S. Printsevskaya, O. V. Miroshnikova, M. I. Reznikova, Maria N. Preobrazhenskaya. Antiretroviral Activity of Semisynthetic Derivatives of Glycopeptide Antibiotics. J. Med. Chem., 2003, 46, 2755-2764
  116.     Jan Balzarini, Christophe Pannecouque, Erik De Clercq, Andrey Y. Pavlov, Svetlana S. Printsevskaya, Olga V. Miroshnikova, Marina I. Reznikova, and Maria N. Preobrazhenskaya Antiretroviral Activity of Semisynthetic Derivatives of Glycopeptide Antibiotics J. Med. Chem., 2003, 46 (13), 2755-2764
  117.     Svetlana S. Printsevskaya, Andrey Y. Pavlov, Evgenia N. Olsufyeva, Elena P. Mirchink, and Maria N. Preobrazhenskaya The role of the glycopeptide framework in the antibacterial activity of hydrophobic derivatives of glycopeptide antibiotics J. Med. Chem. 2003, 46 (7) 1204-1209
  118.     S. S. Printsevskaya, A.Y. Pavlov, E. N. Olsufyeva, E. P. Mirchink, E. B. Isakova, M. I. Reznikova, R. C. Goldman, A.A. Branstrom, E.R. Baizman, C. B. Longley, G. Batta and M. N. Preobrazhenskaya. Synthesis and Mode of Action of Hydrophobic Derivatives of the Glycopeptide Antibiotic Eremomycin and De-(N-methyl-D-leucyl)eremomycin Against Glycopeptide-Sensitive and Resistant Bacteria. J. Med. Chem.2002, 45, 1340-1347
  119.     Svetlana S. Printsevskaya Andrey Y. Pavlov, Evgenia N. Olsufyeva, Elena P. Mirchink, Elena B. Isakova, Marina I. Reznikova, Robert C. Goldman, Arthur A. Branstrom, Eugene R. Baizman, Clifford B. Longley, Gyula Batta and Maria N. Preobrazhenskaya Synthesis and Mode of Action of Hydrophobic Derivatives of the Glycopeptide Antibiotic Eremomycin and De-(N-methyl-D-leucyl)eremomycin Against Glycopeptide-Sensitive and Resistant Bacteria J. Med. Chem.2002, 45, # 6, 1340-1347
  120.     Olga V. Leontieva, Maria N. Preobrazhenskaya, and Ralph J. Bernacki Partial circumvention of P-glycoprotein-mediated multidrug resistance by doxorubicin 14-O-hemiadipate Investigational New Drugs, 20, 35-49 (2002)
  121.     Павлов А.Ю., Принцевская С.С., Олcуфьева Е.Н., и Преображенская М.Н. Полусинтетические производные гликопептидного антибиотика эремомицина , активные в отношении гликопептидорезистентных энтерококков Клиническая микробиология и антимикробная химиотерапия № 3, 2001, Приложение 1, стр. 30
  122.     A.Pavlov, O. Miroshnikova, S. Printsevskaya, E. Olsufyeva, M.Preobrazhenskaya, R. Goldman, A. Branstrom, E. Baizman, C. Longley Synthesis of hydrophobic N'-mono- and N',N''-double alkylated eremomycins inhibiting the trans-glycosylation stage of bacterial cell wall biosynthesis J. Antibiotics 54, No 5, 455 – 459 (2001)
  123.     F. Sztaricskai, G. Batta, Z. Dinya, O. Miroshnikova, M. Preobrazhenskaya, F. Hernadi, A. Koncz, Z. Boda Chemical modification of the eremomycin antibiotic. Formation of a cyclic covalent dimer J. Antibiotics 54, No 3, pp. 314 – 319 (2001)
  124.     О.А. Миргородская*, Е.Н.Олсуфьева**, Д.Е.Колуме, Т.Д.Д. Йоргенсен, П. Роепсторфф, А.Ю.Павлов**, О.В.Мирошникова**, М.Н.Преображенская. Изучение димеризации полусинтетических производных эремомицина методом ESI MS и ее роли в проявлении антибактери-альной активности. Биоорг. Хим. 2000, 26, # 8, 631-640
  125.     О.А. Миргородская*, Е.Н.Олсуфьева**, Д.Е.Колуме, Т.Д.Д. Йоргенсен, П. Роепсторфф, А.Ю.Павлов**, О.В.Мирошникова**, М.Н.Преображенская. Изучение димеризации полусинтетических производных эремомицина методом ESI MS и ее роли в проявлении антибактери-альной активности. Биоорг. Хим. 2000, 26, # 8, 631-640
  126.     O.V. Miroshnikova, S. S. Printsevskaya, E. N. Olsufyeva, A.Y. Pavlov, A. Nilius, D. Hensey-Rudloff and M. N.Preobrazhenskayaa Structure-Activity Relationships in the Series of Eremomycin Carboxamides. J. Antibiotics, 2000, v. 53, 286-293
  127.     О.А.Миргородская, Е.Н.Олсуфьева, Д.Е.Колуме, Т.Д.Д. Йоргенсен, П. Роепсторфф, А.Ю.Павлов, О.В.Мирошникова, М.Н.Преображенская Изучение димеризации полусинтетических производных эремомицина методом ESI MS и ее роли в проявлении антибактериальной активности. Биоорг. Хим. 2000, 26, # 8, 631-640
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  195.     Sergey N. Lavrenov,Yuriy N. Luzikov,Evgeniy E. Bykov,Marina I. Reznikova,Valeria A. Glazunova,Alexander A. Shtil, and Maria N. Preobrazhenskaya Synthesis and Cytotoxic Potency of Novel Tris(1-alkylindol-3-yl)methylium Salts: Role of N-alkyl Substituents Bioorganic & Medicinal Chemistry 18 (2010) 6905–6913
  196.     Hanh H. Nguyen, Sergey N. Lavrenov, Shyam N. Sundar, David H.H. Nguyen , Min Tseng , Crystal N. Marconett , Jenny Kung, Richard E. Staub b, Maria N. Preobrazhenskaya, Leonard F. Bjeldanes, and Gary L. Firestone, 1-Benzyl-indole-3-carbinol is a novel indole-3-carbinol derivative with significantly enhanced potency of anti-proliferative and anti-estrogenic properties in human breast cancer cells Chemico-Biological Interactions Volume 186, Issue 3, 5 August 2010, Pages 255-266
  197.     А.М.Королев,Ю.Н.Лузиков,М.И. Резникова,М.Н.Преображенская 3-O-и 2-С алкилирование солей L-аскорбиновой кислоты бензилгалогенидами и производными N-замещенных индолметанолов ИЗВАН серия химическая 2010, 201, №2, 447-452
  198.     Е.Е.Быков, С.Н.Лавренов, М.Н.Преображенская Квантовохимическое исследование зависимости pKa от рассчитанной энергии отрыва протона для некоторых производных индола и фенола. Химия гетероциклических соединений, 2006, №1 с.47-50
  199.     S. N. Lavrenov, K.F. Turchin, A.M. Korolev, Olga S. Anisimova and Maria N. Preobrazhenskaya. New pyrano[3,4-b]indoles from 2-hydroxymethyl-indole and L-dehydroascorbic acid. Tetrahedron, 2005, V. 61, 6610-6613
  200.     S.N. Lavrenov, N. P. Solovyeva, M.I. Reznikova, O.S. Anisimova, and M.N. Preobrazhenskaya. The interaction of per-o-acetylated acyclic 1-(1-butylindol-3-yl)-1-deoxy-ketoses with silylated uracil. Nucleosides, Nucleotides & Nucleic Acids Vol. 23, N1&2, pp281-289 (2004)
  201.     A. M. Korolev, A. E. Shchekotikhin, L. N. Lysenkova, and M. N. Preobrazhenskaya. Synthesis of (Indol-3-yl)methanesulfonamide and its 5-Methoxy Derivative. Synthesis 2003, # 3, 383-388.
  202.     S.N. Lavrenov, A.M. Korolev, M.I. Reznikova, A.V. Sosnov and M.N. Preobrazhenskaya. Study of 1-deoxy-1-(indol-3-yl)-L-sorbose, 1-deoxy-1-(indol-3-yl)-L-tagatose and their analogs. Carb. Res. V. 338, # 2, 143-152 (2003)
  203.     S.N. Lavrenov, S. A. Lakatosh, L. N. Lysenkova, A. M. Korolev, M. N. Preobrazhenskaya. Synthesis of Methyl 6-and 5-Nitroindole-2-carboxylates by Nitration of Indoline-2-carboxylates. Synthesis 2002, # 3: 320-322
  204.     Л. Н. Лысенкова, М. И. Резникова, А. М. Королев и М. Н. Преображенская. Изучение превращений 2-с-[(индол-3-ил) метил]- -l-ксило-гекс-3-улофуранозо-новой кислоты (от-крытой формы аскорбигена) в кислой среде. Изв. РАН, серия химическая 2001, № 7, 1248-1252
  205.     S.N. Lavrenov, A.M. Korolev and M.N. Preobrazhenskaya. O-Glycosides of N-hydroxyindoles. Nucleosides, Nucleotides & Nucleic acids 2001, 20, #10-11, 1881-1889
  206.     A. M. Korolev, L. N. Yudina, I. I. Rozhkov, L.N. Lysenkova, E. I. Lazhko, Y. N. Luzikov, and M. N. Preobrazhenskaya. The formation of 2-hydroxy-4-hydroxymethyl-3-(indol-3-yl)cyclopent-2-enone derivatives from ascorbigens. Carbohydrate Research. V.330, # 4, pp 469 - 477. (2001)
  207.     M. I. Reznikova, A. M. Korolev, D. A. Bodyagin and M. N. Preobrazhenskaya. Transformations of ascorbigen in vivo into ascorbigen acid and 1-deoxy-1-(indol-3-yl)ketoses. Food Chemistry. 71(4), 469-474 (2000)
  208.     М. Н Преображенская, А. М Королев. Indole Derivatives in Vegetables of the Cruciferae Family. A review. Russian Journal of Bioorganic Chemistry. 2000, 26, 85-97
  209.     M. Preobrazhenskaya*, I. Rozhkov, E. Lazhko, A. Korolev. Interaction of L-Ascorbic acid with DL-N-methyl-?-hydroxytryptamine. Tetrahedron letters, 39, No 1, 109-112, 1998
  210.     I.I.Rozhkov, E.I.Lazhko,L.N.Yudina, A.M.Korolev Reaction of Vanilmandelic acid and 4-hydroxybenzylalcohol derivatives with L- ascorbic acid Tetrahedron Vol. 53, No. 20, 6971-6976, 1997 Corrigendum: Tetrahedron, 55 (1999) 1517
  211.     Ватлин А.А., Беккер О.Б., Лысенкова Л.Н., Королев А.М., Щекотихин А.Е., Даниленко В.Н. Секвенирование и анализ резистома Streptomyces fradiae ATCC 19609 c целью разработки тест-системы для скрининга новых антибактериальных систем. Генетика. 2016 Т.52, №6, С.723-727.
  212.     Tevyashova A.N., Korolev A.M., Trenin A.S., Dezhenkova L.G., Shtil A.A., Polshakov V.I., Savelyev O.Y., Olsufyeva E.N. New conjugates of polyene macrolide amphotericin B with benzoxaboroles: synthesis and properties. J. Antibiotics. 2016. V.69, P. 549-560.
  213.     Лысенкова Л.Н., Савельев О.Ю., Королев А.М., Даниленко В.Н., Беккер О.Б., Мавлетова Д.А., Ватлин А.А., Омельчук О.А., Щекотихин А.Е.. Синтез 33-(R,S)-бромо-33-дезоксиолигомицина А. Макрогетероциклы. 2016, Т.9, №3, С.307-313.
  214.     Lysenkova L.N., Godovikov I.A., Korolev A.M., Danilenko V.N., Bekker O.B., Mavletova D.A., Vatlin A.A., Shchekotikhin A.E., Preobrazhenskaya M.N. Synthesis and anti-actinomycotic activity of the thiocyanato derivative of oligomycin A modified in the 2-hydroxypropyl side chain. Macroheterocyles, 2015, V.8, № 4, doi: 10.6060/mhc151084s.
  215.     Vatlin A.A., Bekker O.B., Lysenkova L.N., Danilenko V.N. Draft Genome Sequence of Streptomyces fradiae olg1-1, a Strain Resistant to Nitrone-Oligomycin. Genome Announcements, 2015 Sep-Oct; 3(5): e01252-15. doi: 10.1128/genomeA.01252-15.
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  220.     Cogoi S., Shchekotikhin A.E., Xodo L.E. HRAS is silenced by two neighboring G-quadruplexesand activated by MAZ, a zinc-finger transcription factor with DNA unfolding property. Nucleic Acids Research, 2014, 42 (13), pp. 8379–8388
  221.     L.N. Lysenkova, K.F. Turchin, A.M. Korolev, V.N Danilenko, O.B Bekker, L.G Dezhenkova, A.A. Shtil, M.N Preobrazhenskaya. Study on retroaldol degradation products of antibiotic oligomycin A. The Journal of Antibiotics (2014) 67, 153–158. (Tokyo). doi:10.1038/ja.2013.92.
  222.     Ol’khovich., Sharapova A.V., Lavrenov S.N., Blokhina S.V., Perlovich G. L. Inclusion complexes of hydroxypropyl-b-cyclodextrin with novel cytotoxic compounds: Solubility and thermodynamic properties. Fluid Phase Equilibria 2014, vol. 384, p. 68–72. (IF = 2.241) WOS
  223.     Lysenkova LN, Turchin KF, Korolev AM,Danilenko VN, Bekker OB, Dezhenkova LG,Shtil AA, Preobrazhenskaya MN. Study on retroaldol degradation products of antibiotic oligomycin A.J Antibiot (Tokyo). doi: 10.1038/ja.2013.92
  224.     Lysenkova LN, Turchin KF, Korolev AM, Dezhenkova LG, Bekker OB, Shtil AA, Danilenko VN, Preobrazhenskaya MN. Synthesis and cytotoxicity of oligomycin A derivatives modified in the side chain. Bioorg Med Chem. (2013)1;21(11):2918-24
  225.     Lapa GB, Bekker OB, Mirchink EP, Danilenko VN, Preobrazhenskaya MN Regioselective acylation of congeners of 3-amino-1H-pyrazolo[3,4-b]quinolines, their activity on bacterial serine/threonine protein kinases and in vitro antibacterial (including antimycobacterial) activity. J Enzyme Inhib Med Chem. 2013 Oct;28(5):1088-93, ИФ-1,495
  226.     J. Schaefer, S.J. Kim, M. Singh, M. Preobrazhenskaya. Staphylococcus aureus Peptidoglycan Stem Packing by Rotational-Echo Double Resonance NMR Spectroscopy. Biochemistry,(2013) v 52, 3651-59
  227.     Lyudmila N Lysenkova, Konstantin F Turchin, Alexander M Korolev, Evgenyi E Bykov, Valery N Danilenko, Olga B Bekker, Alexey S Trenin, Sergei M Elizarov, Lyubov G Dezhenkova, Alexander A Shtil and Maria N Preobrazhenskaya. A novel acyclic oligomycin A derivative formed via retro-aldol rearrangement of oligomycin A. The Journal of Antibiotics (2012) 65, 405–411
  228.     Lyudmila N. Lysenkova1, Konstantin F. Turchin1, Valery N. Danilenko2, Alexander M. Korolev1, and Maria N. Preobrazhenskaya1 The first examples of chemical modification of oligomycin A. The Journal of Antibiotics (2010) 63, 17–22.
  229.     Anna N. Tevyashovaa, Eugenia N. Olsufyevaa, Jan Balzarini, Alexander A. Shtilc, Lyubov G. Dezhenkovac, lLadimir M. Bukhmana, Victor b. Zbarsky, Maria n. Preobrazhenskayaa* Modification of the antibiotic Olivomycin I at the 2’-Keto Group of the Side Chain. Novel Derivatives, Antitumor and Topoisomerase I Poisoning Activity. The Journal of Antibiotics (2009) 62, 37–41
  230.     Maria N. Preobrazhenskaya, Evgenia N. Olsufyeva, Svetlana E. Solovieva, Anna N. Tevyashova,Marina I. Reznikova, Yuryi N. Luzikov, Larisa P. Terekhova, Aleksei S. Trenin, Olga A. Galatenko, Ivan D. Treshalin, Elena P. Mirchink, Vladimir M. Bukhman, Ha#vard Sletta, and Sergey B. Zotchev. Chemical modification and biological evaluation of new semi-synthetic derivatives of S44HP, a genetically engineered anti-fungal polyene macrolide antibiotic, J. Med. Chem., 2009, 52 (1), 189-196
  231.     I. S. Severina, N.V. Pyatakova, A. B. Postnikov, M.N. Preobrazhenskaya, Y. V. Khropov. Antitumour antibiotic streptonigrin and its derivatives as the inhibitors of nitric oxide-dependent activation of soluble guanylate cyclase. European Journal of Pharmacology, 483 (2004), 127-132.
  232.     I. S. Severina, N.V. Pyatakova, A. B. Postnikov, M.N. Preobrazhenskaya, Y. V. Khropov. Antitumour antibiotic streptonigrin and its derivatives as the inhibitors of nitric oxide-dependent activation of soluble guanylate cyclase. European Journal of Pharmacology, 483 (2004), 127-132.
  233.     N.V.Holpne-Kozlova, E.I.Lazhko and M.N. Preobrazhenskaya.Transformation of streptonigrin into streptonigrone and biological evaluation of antibiotic streptonigrin and streptonigrone alkyl ethers. J.Antibiotics, v.45, N 2, p.227-234,1992
  234.     V.V.Tolstikov,J.Balzarini, E.De Clercq and M.N. Preobrazhenskaya. Chemical modification of antibiotic streptonigrin: Synthesis and properties of 2-decarboxy-2-amino- streptonigrin (streptonigrone-imine) J.Antibiotics, 1992, v.45, N 6, p.1002-1007
  235.     V.V.Tolstikov, T.D.Oreshkina, T.V.Osipova, F.Sztarickai, J.Balzarini, E.De Clercq, N.V.Holpne-Kozlova M.N.Preobrazhenskaya. Amides of antibiotic streptonigrin and aminodicarboxylic acids or aminosugars, synthesis and biological evaluation. J.Antibiotics, 1992 v.45,N 6, p.1020-1025

 

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